Inaperisone

Inaperisone
Clinical data

ATC code	None
Identifiers
IUPAC name 1-(4-Ethylphenyl)-2-methyl-3-(1-pyrrolidinyl)-1-propanone
CAS Number	99323-21-4
PubChem (CID)	65860
ChemSpider	59271
ChEMBL	CHEMBL1797127
Chemical and physical data
Formula	C₁₆H₂₃NO
Molar mass	245.360 g/mol
3D model (Jmol)	Interactive image
SMILES CCC1=CC=C(C=C1)C(=O)C(C)CN2CCCC2
InChI InChI=1S/C16H23NO/c1-3-14-6-8-15(9-7-14)16(18)13(2)12-17-10-4-5-11-17/h6-9,13H,3-5,10-12H2,1-2H3 Key:VNFAARJCGSAROU-UHFFFAOYSA-N

Inaperisone (INN) is a muscle relaxant.^[1]

See also

Chemically and mechanistically related drugs: eperisone, lanperisone, silperisone, tolperisone

References

↑ Nagata, O.; Murata, M.; Kato, H.; Terasaki, T.; Sato, H.; Tsuji, A. (1990). "Physiological pharmacokinetics of a new muscle-relaxant, inaperisone, combined with its pharmacological effect on blood flow rate". Drug metabolism and disposition: the biological fate of chemicals. 18 (6): 902–910. PMID 1981535.

Skeletal muscle relaxants (M03)

Peripherally acting
(primarily antinicotinic,
NMJ block)

Non-depolarizing

Curare alkaloids	Alcuronium Dimethyltubocurarine Tubocurarine

4° ammonium agents	ultra-short duration: Gantacurium short duration: Mivacurium Chandonium intermediate duration: Atracurium Cisatracurium Fazadinium Rocuronium Vecuronium long duration: Doxacurium Dimethyltubocurarine Pancuronium Pipecuronium Laudexium Gallamine unsorted: Hexafluronium (Hexafluorenium)

Choline derivatives: Suxamethonium (Succinylcholine)

Polyalkylene derivatives: Hexamethonium

ACh release inhibitors

Botulinum toxin

Centrally acting

Carbamic acid esters	Carisoprodol Cyclarbamate Difebarbamate Febarbamate Meprobamate Phenprobamate Styramate Tybamate

Benzodiazepines	Bromazepam Diazepam Clonazepam Flunitrazepam Lorazepam Nitrazepam Temazepam Tetrazepam

Nonbenzodiazepines	Eszopiclone

Thienodiazepines	Etizolam

Quinazolines	Methaqualone

Anticholinergics (Antimuscarinics)	Cyclobenzaprine Orphenadrine

Other	Arbaclofen placarbil Baclofen Chlormezanone Chlorphenesin Chlorzoxazone Donepezil Eperisone Fenyramidol Flopropione Gabapentin GHB Inaperisone Lanperisone Mephenesin Mephenoxalone Metaxalone Methocarbamol Phenibut Pregabalin Pridinol Promoxolane Quinine Silperisone Thiocolchicoside Tizanidine Tolperisone Zoxazolamine

Directly acting

Dantrolene

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