Rimazolium

Rimazolium
Clinical data

ATC code	N02BG02 (WHO)
Identifiers
IUPAC name 3-(Ethoxycarbonyl)-1,6-dimethyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-1-ium
CAS Number	35615-72-6 28610-84-6 (mesylate)
PubChem (CID)	71940
ChemSpider	64949
ECHA InfoCard	100.047.844
Chemical and physical data
Formula	C₁₃H₁₉N₂O₃ C₁₄H₂₂N₂O₇S (mesylate)
Molar mass	251.30 g/mol 362.40 g/mol (mesylate)
3D model (Jmol)	Interactive image
Melting point	165 to 166 °C (329 to 331 °F) (mesylate)^[1]
SMILES O=C1C(=C/[N+](=C2\N1C(CCC2)C)C)\C(=O)OCC
InChI InChI=1S/C13H19N2O3/c1-4-18-13(17)10-8-14(3)11-7-5-6-9(2)15(11)12(10)16/h8-9H,4-7H2,1-3H3/q+1 Key:JOWRFSPJFXLGGY-UHFFFAOYSA-N

Rimazolium is a non-narcotic analgesic.^[1]^[2] It is usually formulated as the mesylate salt, rimazolium metilsufate.

References

1 2 Merck Index, 11th Edition, 8222
↑ Furst, S; Gyires, K; Knoll, J (1988). "Analgesic profile of rimazolium as compared to different classes of pain killers". Arzneimittel-Forschung. 38 (4): 552–7. PMID 3261171.

Opiates/opium	Codeine^# (+paracetamol, +aspirin) Morphine^# (+naltrexone) Opium Laudanum Paregoric

Semisynthetic	Acetyldihydrocodeine Benzylmorphine Buprenorphine (+naloxone) Desomorphine Diamorphine (heroin) Dihydrocodeine (+paracetamol) Dihydromorphine Ethylmorphine Hydrocodone (+paracetamol, +ibuprofen, +aspirin) Hydromorphinol Hydromorphone Nicocodeine Nicodicodeine Nicomorphine Oxycodone (+paracetamol, +aspirin, +ibuprofen, +naloxone, +naltrexone) Oxymorphone Thebacon

Synthetic	Alphaprodine Anileridine Butorphanol Dextromoramide Dextropropoxyphene Dezocine Fentanyl (+fluanisone) Ketobemidone Levorphanol Meptazinol Methadone Nalbuphine Pentazocine Pethidine Phenadoxone Phenazocine Piminodine Piritramide Propiram Tapentadol Tilidine Tramadol

Propionates	Fenoprofen Flurbiprofen Ibuprofen^# Ketoprofen Naproxen Oxaprozin

Oxicams	Meloxicam Piroxicam

Acetates	Diclofenac Indometacin Ketorolac Nabumetone Sulindac Tolmetin

COX-2 inhibitors	Celecoxib Etoricoxib Lumiracoxib Parecoxib Rofecoxib ^‡ Valdecoxib ^‡

Fenamates	Meclofenamic acid Mefenamic acid

Salicylates	Aspirin (acetylsalicylic acid)^# (+paracetamol/caffeine) Benorylate Diflunisal Ethenzamide Magnesium salicylate Salicin Salicylamide Salsalate Wintergreen (methyl salicylate)

Pyrazolones	Aminophenazone^‡ Ampyrone Metamizole (dipyrone) Nifenazone Phenazone Propyphenazone

Others	Glafenine

Calcium blockers	Gabapentin Gabapentin enacarbil Pregabalin Ziconotide

Sodium blockers	Carbamazepine Lacosamide Local anesthetics (e.g., cocaine, lidocaine) Mexiletine Nefopam Tricyclic antidepressants (e.g., amitriptyline^#) Na_v1.7/1.8-selective: DSP-2230^§ Funapide^§ PF-05089771^§ Raxatrigine^§

Potassium openers	Flupirtine

Others

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