Chlorphenoxamine
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| Clinical data | |
|---|---|
| AHFS/Drugs.com | International Drug Names |
| Routes of administration | Oral, topical |
| ATC code | D04AA34 (WHO) R06AA06 (WHO) |
| Pharmacokinetic data | |
| Bioavailability | Well absorbed |
| Metabolism | Likely hepatic |
| Excretion | Renal |
| Identifiers | |
| |
| CAS Number |
77-38-3 |
| PubChem (CID) | 6475 |
| DrugBank |
DB09007 |
| ChemSpider |
6230 |
| UNII |
3UVD77BP8R |
| KEGG |
D07198 |
| ChEMBL |
CHEMBL2110774 |
| ECHA InfoCard | 100.115.538 |
| Chemical and physical data | |
| Formula | C18H22ClNO |
| Molar mass | 303.826 g/mol |
| 3D model (Jmol) | Interactive image |
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Chlorphenoxamine (Phenoxene) is an antihistamine and anticholinergic used as an antipruritic[1] and antiparkinsonian[2] agent. It is an analog of diphenhydramine.[3]
References
- ↑ Bazex, A.; Dupre, A.; Christol, B. (1963). "Trial treatment of urticaria with chlorphenoxamine". Clinique (Paris, France). 58: 447–450. PMID 13967113.
- ↑ Uldall, P. R.; Walton, J. N.; Newell, D. J. (1961). "Chlorphenoxamine hydrochloride in parkinsonism. A controlled trial". British Medical Journal. 1 (5240): 1649–1652. doi:10.1136/bmj.1.5240.1649. PMC 1954253
. PMID 13779077. - ↑ H. Arnold, N. Brock, E. Kuhas, and D. Lorenz, Arzneimittel Forsch., 4, 189 (1954).
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